Bioheterocycles 2019

Programme

Click on the day below to see the detailed programme.
Monday 17/06/2019
08:00Registration
09:10Opening
Prof. Matthias D'HOOGHE
(GHENT UNIVERSITY, Ghent, Belgium)
Session 1
Session Chair
Prof. Christian STEVENS
(UGENT, Ghent, Belgium)
09:30Heterocycles as Key Features of New Starting Points for Drug Discovery (PL01)
Dr Peter MEIER
(NOVARTIS PHARMA AG, Basel, Switzerland)
10:15Development of Enzyme Inhibitors and Multi-target-directed Ligands for Treating Neurodegenerative Diseases (IL01)
Prof. Stanislav GOBEC
(UNIVERSITY OF LJUBLJANA, Ljubljana, Slovenia)
10:45Coffee break
Session 2
Session Chair
Prof. Till OPATZ
(JOHANNES GUTENBERG-UNIVERSITY, Mainz, Germany)
11:15Silil-Prins Cyclization: Towards the Synthesis of Medium Sized Heterocycles (OC01)
Prof. Asuncion BARBERO
(UNIVERSITY OF VALLADOLID, Valladolid, Spain)
11:30Chiral Piperidines from Pyridines: the Meta-Substitution Challenge in Asymmetric Hydrogenation (OC02)
Dr Paul ALSTERS
(INNOSYN B.V., Geleen, The Netherlands)
11:45Expanding the Chemical Space of Chiral Trifunctional Building Blocks by Stereoselective Synthesis from Natural Terpenes (IL02)
Prof. Zsolt SZAKONYI
(UNIVERSITY OF SZEGED, Szeged, Hungary)
12:15Lunch
Session 3
Session Chair
Prof. Fawaz ALDABBAGH
(KINGSTON UNIVERSITY, London, United Kingdom)
13:30A Journey in Heteroaromatic Scaffolds as Protein Kinase Inhibitors (PL02)
Prof. Pascale MOREAU
(UNIVERSITY OF CLERMONT AUVERGNE, Aubière, France)
14:15Bacterial Quinolones and Derivatives: New Drugs for Bad Bugs (IL03)
Dr Thomas BOTTCHER
(UNIVERSITY OF KONSTANZ, Konstanz, Germany)
14:45Hydrogen Peroxide and Hydrohalic Acid-Mediated Synthesis of Ring-Fused Benzimidazolequinone Anti-Cancer Agents (OC03)
Mr Darren CONBOY
(KINGSTON UNIVERSITY LONDON, Kingston upon Thames, United Kingdom)
15:00Coffee break
Session 4
Session Chair
Dr Bart ROMAN
(GHENT UNIVERSITY, Ghent, Belgium)
15:30Thionations Using a P4S10-Pyridine Complex (OC04)
Ms Ngarita KINGI
(VIRONOVA MEDICAL AB, Stockholm, Sweden)
15:45First Solid-Phase Strategy for the Total Synthesis of Fengycin Derivatives, a Class of Cyclic Lipodepsipeptides (OC05)
Dr Lidia FELIU
(LIPPSO, UNIVERSITY OF GIRONA, Girona, Spain)
16:00Design and Synthesis of New Nitrogen-Containing Heterocycles for the Treatment of Mechanical Allodynia (OC06)
Ms Alexia VISSEQ
(INSTITUT DE CHIMIE DE CLERMONT FERRAND, AUBIERE, France)
16:15Poster Session
18:00Welcome Reception (Ghent City Hall)
Tuesday 18/06/2019
Session 5
Session Chair
Prof. Bert MAES
(UNIVERSITY OF ANTWERP, Antwerp, Belgium)
09:00Heterocycles To Control Immune Cell Function (PL03)
Prof. David FAIRLIE
(UNIVERSITY OF QUEENSLAND, Brisbane, Australia)
09:45Vitamin B12 – an Intriguing Bioheterocycle (IL04)
Prof. Dorota GRYKO
(INSTITUTE OF ORGANIC CHEMISTRY PAS, Warsaw, Poland)
10:15Hydroxylated Heterocycles as a Bioisosteric Tool to Modulate the Carboxylic Function (OC08)
Dr Agnese Chiara PIPPIONE
(UNIVERSITY OF TURIN, Torino, Italy)
10:30Tweaking the Blebbistatin Scaffold Towards Better Pharmacological Tools (OC09)
Dr Bart ROMAN
(GHENT UNIVERSITY, Ghent, Belgium)
10:45Coffee break
Session 6
Session Chair
Prof. Asuncion BARBERO
(UNIVERSITY OF VALLADOLID, Valladolid, Spain)
11:15The Magic of Wood and Light – New Concepts for Synthetic Chemistry (OC10)
Prof. Till OPATZ
(JOHANNES GUTENBERG-UNIVERSITY, Mainz, Germany)
11:30Synthesis of Enantioenriched 3-Isobenzofuranones Using Chiral Organomagnesiates (OC11)
Dr Sabrina TOUCHET
(UNIVERSITÉ DE LORRAINE, Vandoeuvre-les-Nancy, France)
11:45Functionalization of Aromatic Heterocycles Using Bases Derived from LiTMP (IL05)
Prof. Florence MONGIN
(UNIVERSITY OF RENNES, Rennes, France)
12:15Lunch
Session 7
Session Chair
Prof. Stanislav GOBEC
(UNIVERSITY OF LJUBLJANA, Ljubljana, Slovenia)
13:30Synthesis of Heterocyles Using Visible Light Photocatalysis (PL04)
Prof. Burkhard KÖNIG
(UNIVERSITY OF REGENSBURG, Regensburg, Germany)
14:15Leveraging Carbonylation and N-acyl imine Chemistry in Heterocycle Synthesis (IL06)
Dr Luke ODELL
(UNIVERSITY OF UPPSALA, Uppsala, Sweden)
14:45Structurally Simple Cytosine Peptidomimetics as Potent Cardioprotectors in Myocardial Ischemia (MI) Mouse Model: Design, Synthesis And Biological Evaluation (OC12)
Dr Edward KORSHIN
(BAR-ILAN UNIVERSITY, Ramat Gan, Israel)
15:00Biradical Formation by Deprotonation in Conjugated 2-Amino/Imino Thiazole Derivatives (OC13)
Prof. Francisco LOPEZ-CALAHORRA
(UNIVERSITAT DE BARCELONA, Barcelona, Spain)
16:00Excursion
Wednesday 19/06/2019
Session 8
Session Chair
Prof. Wim DE BORGGRAEVE
(KU LEUVEN, Leuven, Belgium)
09:00The Beautiful Simplicity of Rearrangements (PL05)
Prof. Nuno MAULIDE
(UNIVERSITY OF VIENNA, Vienna, Austria)
09:45A journey with Saponins (IL07)
Dr Martina LAHMANN
(BANGOR UNIVERSITY, Wales, United Kingdom)
10:15Small but Selective: Developing Chemical Probes for PKN/PRK2 (OC14)
Dr Fiona SCOTT
(SUSSEX DRUG DISCOVERY CENTRE, Falmer, United Kingdom)
10:30Application of Tsunoda reagent to the convenient synthesis of drug-like pyrazoles (OC15)
Dr Olivier LORTHIOIR
(ASTRAZENECA, Cambridge, United Kingdom)
10:45Coffee break
Session 9
Session Chair
Prof. Florence MONGIN
(UNIVERSITY OF RENNES, Rennes, France)
11:15The Phenanthridine PJ-34 Exclusively Eradicates Human cancer Cells (OC16)
Prof. Malka COHEN-ARMON
(TEL-AVIV UNIVERSITY, Tel-Aviv, Israel)
11:30Synthesis and in vitro -Glucosidase Inhibitory Activity of Polyhydroxylated 2-Styrylchromones (OC17)
Dr Clementina SANTOS
(INSTITUTO POLITÉCNICO DE BRAGANÇA, Braganca, Portugal)
11:45Heterocycles and Neglected Diseases: Still a Role for Total Synthesis (IL08)
Prof. Adrian DOBBS
(UNIVERSITY OF GREENWICH, Kent, United Kingdom)
12:15Lunch
Session 10
Session Chair
Prof. Zsolt SZAKONYI
(UNIVERSITY OF SZEGED, Szeged, Hungary)
13:30Multiple Conjugation Reactions on Peptides and Oligonucleotides (PL06)
Prof. Anna GRANDAS
(UNIVERSITY OF BARCELONA, Barcelona, Spain)
14:15Heterocycles as a Route to New Chemical Space for Drug Discovery (IL09)
Prof. James BULL
(IMPERIAL COLLEGE, London, United Kingdom)
14:45'Stretched' Analogs of Piperidine, Piperazine, and Morpholine: Advanced Building Blocks for Drug Discovery (OC18)
Dr Ivan KONDRATOV
(ENAMINE, Kiev, Ukraine)
15:00Coffee break
Session 11
Session Chair
Dr Thomas HEUGEBAERT
(UGENT, Gent, Belgium)
15:30Biologically Active Oxygen and Nitrogen Heterocyclic Compounds from Cycloaddition and Conjugate Addition Reactions On Chromones (OC19)
Prof. Artur M.S. SILVA
(UNIVERSITY OF AVEIRO, Aveiro, Portugal)
15:45Combining Isocyanides with Carbon Dioxide for Heterocycle Synthesis (OC20)
Mr Jeroen BOMON
(UNIVERSITEIT ANTWERPEN, Antwerpen, Belgium)
16:00Kolbe Anodic Decarboxylation as a Green Way to Access Pyrrolidinones (OC21)
Ms Mathilde QUERTENMONT
(UNIVERSITÉ CATHOLIQUE DE LOUVAIN, La Hulpe, Belgium)
16:15Playing with Properties of Biologically Active Compounds: High-Throughput Conjugation of Drug-Like Molecules for Chemical Biology (OC22)
Ms Sona KRAJCOVICOVA
(PALACKY UNIVERSITY, Olomouc, Czech Republic)
16:30Poster Session
19:00Symposium Banquet
Thursday 20/06/2019
Session 12
Session Chair
Prof. Sven MANGELINCKX
(GHENT UNIVERSITY, Ghent, Belgium)
10:00Heterocyclic Chemistry in Drug Development (PL07)
Prof. Wim DE BORGGRAEVE
(KU LEUVEN, Leuven, Belgium)
10:45Biologically Active Azaheterocycles Containing a Ferrocene Moiety (IL10)
Prof. Niko S. RADULOVIC
(UNIVERSITY OF NIS, Nis, Serbia)
11:15Regioselective C-H Arylation of Nitro Heterocycles and Further Transformation of Manipulable Nitro Group (OC23)
Dr Viktor IAROSHENKO
(POLISH ACADEMY OF SCIENCES, Lodz, Poland)
11:30Towards DNA-Encoded Heterocycle Libraries - DNA-Compatible Povarov and Groebke Reactions by Micellar Broensted Acid Catalysis (OC24)
Dr Andreas BRUNSCHWEIGER
(TU DORTMUND, Dortmund, Germany)
11:45Closing and Award ceremony
Prof. Matthias D'HOOGHE
(GHENT UNIVERSITY, Ghent, Belgium)
12:00Lunch

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