10th EFMC Short Course on Medicinal Chemistry

ONLINE REGISTRATION IS NOW OPEN !
Register now!

Sunday April 12, 2015
18:00Dinner
Monday April 13, 2015
Breakfast (as of 7:30)
08:30Introduction
09:00Nuclear Receptor Protein-Protein Interactions
Prof. Luc BRUNSVELD
(EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands)
10:30Coffee Break
11:00Nuclear Receptor Protein-Protein Interactions - Part II
Prof. Luc BRUNSVELD
(EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands)
12:30Lunch
13:30Stabilization of PPIs: the Other Side of PPI Modulation
Dr Christian OTTMANN
(EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands)
15:30Coffee Break
16:00Stabilization of PPIs: the Other Side of PPI Modulation - Part II
Dr Christian OTTMANN
(EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands)
17:30Day End
Tuesday April 14, 2015
Breakfast (as of 7:30)
08:30Modern Methods for Targeting Low Affinity Protein-Protein Interactions: Structure and Function
Prof. Anna MAPP
(UNIVERSITY OF MICHIGAN, Ann-Arbor, United States)
10:30Coffee Break
11:00Modern Methods for Targeting Low Affinity Protein-Protein Interactions: Structure and Function - Part II
Prof. Anna MAPP
(UNIVERSITY OF MICHIGAN, Ann-Arbor, United States)
12:30Lunch
13:30Design and Synthesis of PPI-focussed Chemical Libraries
Dr Fabrizio GIORDANETTO
(TAROS CHEMICALS, New York, United States)
15:30Coffee Break
16:00Design and Evaluation of Biophysical Assays for the Identification of PPI-Modulators
Dr Alexander WOLF
(LEAD DISCOVERY, Dortmund, Germany)
17:30Day End
Wednesday April 15, 2015
Breakfast (as of 7:30)
08:30Developing Small Molecule Inhibitors of Bromodomain-Based Protein-Protein Interactions
Prof. Stuart CONWAY
(UNIVERSITY OF OXFORD, Oxford, United Kingdom)
10:30Coffee Break
11:00Structure-Based Guided Development & Experimental Validation of a Focused Chemical Library Dedicated to Orthosteric Modulation of Protein-Protein Interactions
Dr Xavier MORELLI
(CNRS, MARSEILLE CEDEX 9, France)
12:30Wrap up and Lunch

Copyright 2018 LD Organisation  |  rue Michel de Ghelderode 33/02 B-1348  Louvain-la-Neuve (Belgium)  Tel. +32 10 454777  |   |  VAT: BE 0464819842
Developed and powered by Antalys