Modulation of Enzymes; Epigenetics and Beyond
Oegstgeest (near Leiden), The Netherlands April 24-27, 2016
Breakfast
Introduction
Coffee Break
Epigenetic Target Families in Medicinal Chemistry
Prof. Paul BRENNAN
UNIVERSITY OF OXFORD, Oxford, United Kingdom
Lunch
BETting on Epigenetic Targets: From Phenotypic Discovery to First Time in Man
Dr Chun-wa CHUNG
GLAXOSMITHKLINE R&D, Stevenage, United Kingdom
Coffee Break
Hands on Tutorial - Case Study I: Development of a Kinase Inhibitor
Dr Leon VAN BERKOM
MERCACHEM-SYNCOM, Nijmegen, The Netherlands
Day End
Breakfast
Coffee Break
Lunch
Glycomimetics - an Underexplored Compound Class for Medicinal Chemistry
Prof. Dr Beat ERNST
UNIVERSITY OF BASEL, Basel, Switzerland
Coffee Break
Hands on Tutorial - Case Study II: Development of a HIV Medicine
Dr Stijn GREMMEN
MERCACHEM, Nijmegen, The Netherlands
Day End