Breakfast

Introduction

Protein Kinase Inhibitors

Dr Gerhard MÜLLER
MERCACHEM, Martinsried, Germany

Coffee Break

Epigenetic Target Families in Medicinal Chemistry

Prof. Paul BRENNAN
UNIVERSITY OF OXFORD, Oxford, United Kingdom

Lunch

BETting on Epigenetic Targets: From Phenotypic Discovery to First Time in Man

Dr Chun-wa CHUNG
GLAXOSMITHKLINE R&D, Stevenage, United Kingdom

Coffee Break

Hands on Tutorial - Case Study I: Development of a Kinase Inhibitor

Dr Leon VAN BERKOM
MERCACHEM-SYNCOM, Nijmegen, The Netherlands

Day End

Breakfast

Proteases as Drug Targets

Dr Holger SELLNER
NOVARTIS PHARMA AG, Basel, Switzerland

Coffee Break

Proteasome Inhibitors

Prof. Michael GROLL
TECHNISCHE UNIVERSITÄT MÜNCHEN, Garching, Germany

Lunch

Glycomimetics - an Underexplored Compound Class for Medicinal Chemistry

Prof. Dr Beat ERNST
UNIVERSITY OF BASEL, Basel, Switzerland

Coffee Break

Hands on Tutorial - Case Study II: Development of a HIV Medicine

Dr Stijn GREMMEN
MERCACHEM, Nijmegen, The Netherlands

Day End

Breakfast

The PDE Family and Inhibitors

Dr Andrew BELL
IMPERIAL COLLEGE LONDON, London, United Kingdom

Coffee break

Fragment-Based Lead Generation

Prof. Iwan DE ESCH
VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands

Wrap-up and Lunch