LD Organisation

Scientific Conference Producers

Programme


08:00

Registration

09:15

Welcome Session

Prof. André TARTAR
UNIVERSITY LILLE 2, Lille, France
Prof. Gerald GUILLAUMET
UNIVERSITÉ D'ORLÉANS, Orléans, France

First Session: In Silico Selection

Session Chair:

Prof Luc MORIN-ALLORY
UNIVERSITY OF ORLEANS, Orléans, France

09:30

Navigation in Chemistry Universe Towards Biological Activity

Dr Peter ERTL
NOVARTIS INSTITUTE FOR BIOMEDICAL RESEARCH, Basel, Switzerland

10:15

Structure-Based in Silico Screening: Free Tools and Applications

Dr. Bruno VILLOUTREIX
INSERM - UNIVERSITY PARIS DIDEROT, Paris, France

Second Session: From Target Identification to Development

Session Chair:

Dr Philippe PITCHEN
FOREST RESEARCH INSTITUTE, Hauppauge, United States

11:00

The Therapeutic Potential of Pharmacological Inhibitors of Cyclin-Dependent Kinases

Dr Laurent MEIJER
CNRS - ROSCOFF, Roscoff, France

11:45

Targeted Small Molecule Anti-Cancer Drugs: an Asian Perspective from Discovery to Clinical

Dr. Stéphanie BLANCHARD
S*BIO, Singapore, Singapore

12:30

Lunch and Poster Session

12:30

Career Session in parallel From 12:30 till 16:00

Second Session: From Target Identification to Development (Fol.)

Session Chair:

Dr Luc VAN HIJFTE
JANSSEN CILAG, Val de Reuil, France

14:30

Selective Inhibitors of MMP-12 : from Chemistry to Therapeutic Applications

Dr. Vincent DIVE
CEA, Gif-sur-Yvette, France

15:15

Discovery of the Macrocyclic HCV Protease Inhibitor TMC435350

Dr Pierre RABOISSON
JANSSEN PHARMACEUTICAL COMPANIES

16:00

Coffee Break and Poster Session

Session Chair:

Dr Solo GOLDSTEIN
INSTITUT DE RECHERCHES SERVIER, Suresnes, France

16:30

Irreversible Serine Protease Inhibitors: Useful Tools in Drug Discovery

Prof. Koen AUGUSTYNS
UNIVERSITY OF ANTWERP, Antwerp, Belgium

17:15

« Paul Ehrlich» Lecture: Discovery of Xarelto, a Novel, Oral Antithrombotic Agent

Dr. Susanne ROEHRIG
BAYER SCHERING PHARMA, Wuppertal, Germany

18:00

« Paul Ehrlich» Lecture Award

Prof. Gerald GUILLAUMET
UNIVERSITÉ D'ORLÉANS, Orléans, France
Prof. André TARTAR
UNIVERSITY LILLE 2, Lille, France

19:30

Welcome Cocktail at Hôtel Groslot (Offered by Mr. Serge Grouard, the Mayor of Orléans)

10:30

Start of sessions

Third Session: Interfacing Chembio and Medchem
Fifth Session: Imaging
Third Session: Interfacing Chembio and Medchem
Session Chair:
Prof. Gerard DELERIS
UNIVERSITY BORDEAUX SEGALEN, Bordeaux, France
Fifth Session: Imaging
Session Chair:
Dr. Jean Claude BELOEIL
CNRS UPR 4301, Orléans, France
17:00

Start of sessions

Fourth Session: Synthesis and Lead Optimization
Sixth Session: High Throughput Screening and Lead Identification
Fourth Session: Synthesis and Lead Optimization
Session Chair:
Ing Michel CALDERINI
MERCK, Darmstadt, Germany
Sixth Session: High Throughput Screening and Lead Identification
Session Chair:
Dr Pascal GEORGE
SANOFI-AVENTIS R&D, Longvilliers, France
18:30

End of Conference

18:45

Departure to Gala Dinner

Fourth Session: Synthesis and Lead Optimization (fol.)

Session Chair:

Dr Françoise GUERITTE
INSERM - CNRS, Gif-sur-Yvette, France

09:00

Taking up the Adme Challenge

Prof. Benoit DEPREZ
UNIVERSITY OF LILLE 2, Lille, France

09:45

Discovery of Novel Potent, Selective and Orally Efficacious A2B Adenosine Receptor Antagonists.

Dr. Bernat VIDAL
LABORATORIOS ALMIRALL, Barcelona, Spain

10:30

Coffee Break and Poster Session

Session Chair:

Prof Chris KRUSE
ABBOTT, Weesp, The Netherlands

11:00

New Synthetic Methods and their Application to the Preparation of Biologically Active Molecules

Prof. Mike SHIPMAN
UNIVERSITY OF WARWICK, Coventry, United Kingdom

11:45

« Prix Charles Mentzer »: From Heparin to New Anticoagulants with Unprecedented Pharmacological Profile

Dr. Maurice PETITOU
ENDOTIS PHARMA, Romainville, France

12:30

« Prix Charles Mentzer » Award

Prof. Gerald GUILLAUMET
UNIVERSITÉ D'ORLÉANS, Orléans, France
Prof. André TARTAR
UNIVERSITY LILLE 2, Lille, France

12:35

Lunch and Poster Session

Seventh Session: Biophysics Tools and ADME Tox

Session Chair:

Dr Bruno FIGADERE
UNIVERSITÉ PARIS-SUD, Chatenay-Malabry, France

14:00

Biophysical Approaches in the Hit-to-Lead Optimisation Strategy

Dr. Jean BOUTIN
INSTITUT DE RECHERCHES SERVIER, Croissy-sur-Seine, France

14:45

ADME-PK Optimization Strategies in Drug Discovery and Selection

Dr. Sonia POLI
ADDEX PHARMA, Plan-les-Ouates, Switzerland

15:30

Poster Prizes

16:00

Conclusions

Prof. Gerald GUILLAUMET
UNIVERSITÉ D'ORLÉANS, Orléans, France

Prof. André TARTAR
UNIVERSITY LILLE 2, Lille, France