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Sunday April 28, 2019 |
17:00 | Registration |
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19:00 | Dinner |
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Monday April 29, 2019 |
07:30 | Breakfast |
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08:00 | Opening |
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08:30 | Introduction to Fragment Based Discovery – Overview of the Process and a Historical Perspective |
Prof. Rod HUBBARD (UNIVERSITY OF YORK & VERNALIS, Cambridge, United Kingdom) |
10:30 | Coffee Break |
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11:00 | Design Principles for Fragment Libraries |
Prof. György KESERU (HUNGARIAN ACADEMY OF SCIENCES, Budapest, Hungary) |
12:30 | Lunch |
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13:30 | Experiences and Issues with Biochemical Assays in Fragment-Based Drug Discovery |
Dr Paul ENGLAND (IOTA PHARMACEUTICALS LTD., Cambridge, United Kingdom) |
15:00 | Coffee Break |
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15:30 | Biophysical Fragment Based Screening |
Dr Ben DAVIS (VERNALIS RESEARCH, Cambridge, United Kingdom) |
17:30 | Day End |
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18:00 | Walking tour through Leiden |
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19:00 | Dinner in Leiden |
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Tuesday April 30, 2019 |
07:30 | Breakfast |
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08:30 | Why Fragments Make Sense and Actually Work |
(BIOIB‚RICA) |
10:30 | Coffee Break |
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11:00 | Computational Approaches for Fragment Screening and Fragment Evolution |
Prof. Xavier BARRIL (UNIVERSITY OF BARCELONA & GAIN THERAPEUTICS, Barcelona, Spain) |
12:30 | Lunch |
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13:30 | Applications of FBDD |
Dr Gregg SIEGAL (ZOBIO BV, Leiden, The Netherlands) |
15:00 | Coffee Break |
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15:30 | Application-Project in group (Part 1) |
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17:30 | Day End |
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19:00 | Dinner |
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Wednesday May 1, 2019 |
07:30 | Breakfast |
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08:30 | Application-Project in group (Part 2) |
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10:30 | Coffee Break |
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11:00 | Presentations of the results |
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12:00 | Wrap-up and Lunch |
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