15th EFMC Short Course on Medicinal Chemistry
Sunday April 28, 2019
17:00Registration
19:00Dinner
Monday April 29, 2019
07:30Breakfast
08:00Opening
08:30Introduction to Fragment Based Discovery – Overview of the Process and a Historical Perspective
Prof. Rod HUBBARD
(UNIVERSITY OF YORK & VERNALIS, Cambridge, United Kingdom)
10:30Coffee Break
11:00Design Principles for Fragment Libraries
Prof. György KESERU
(HUNGARIAN ACADEMY OF SCIENCES, Budapest, Hungary)
12:30Lunch
13:30Experiences and Issues with Biochemical Assays in Fragment-Based Drug Discovery
Dr Paul ENGLAND
(IOTA PHARMACEUTICALS LTD., Cambridge, United Kingdom)
15:00Coffee Break
15:30Biophysical Fragment Based Screening
Dr Ben DAVIS
(VERNALIS RESEARCH, Cambridge, United Kingdom)
17:30Day End
18:00Walking tour through Leiden
19:00Dinner in Leiden
Tuesday April 30, 2019
07:30Breakfast
08:30Why Fragments Make Sense and Actually Work

(BIOIB‚RICA)
10:30Coffee Break
11:00Computational Approaches for Fragment Screening and Fragment Evolution
Prof. Xavier BARRIL
(UNIVERSITY OF BARCELONA & GAIN THERAPEUTICS, Barcelona, Spain)
12:30Lunch
13:30Applications of FBDD
Dr Gregg SIEGAL
(ZOBIO BV, Leiden, The Netherlands)
15:00Coffee Break
15:30Application-Project in group (Part 1)
17:30Day End
19:00Dinner
Wednesday May 1, 2019
07:30Breakfast
08:30Application-Project in group (Part 2)
10:30Coffee Break
11:00Presentations of the results
12:00Wrap-up and Lunch

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