Bioheterocycles 2015
Monday June 8, 2015
Session Chair:
Prof. Gilbert KIRSCH
(UNIVERSITÉ DE LORRAINE, Metz, France)
09:00Opening
09:30PL01 - Photoreactive Heterocycles and Natural Product Derivatives
Prof. Dr Thomas LINDEL
(TECHNICAL UNIVERSITY OF BRAUNSCHWEIG, Braunschweig, Germany)
10:25Coffee Break
Session Chair:
Prof. Mercedes ÁLVAREZ
(UNIVERSITY OF BARCELONA, Barcelona, Spain)
10:55PL02 - Targeting DNA Methylation: a Medicinal Chemistry Approach
Prof. Antonello MAI
(UNIVERSITY OF ROME "LA SAPIENZA", Rome, Italy)
11:50IL01 - Synthetic Explorations in Small-ring Azaheterocyclic Chemistry and Development of Novel Bioactive Heterocycles
Prof. Matthias D'HOOGHE
(GHENT UNIVERSITY, Ghent, Belgium)
12:20OC01 - Heterocycle-Peptide Hybrids: Synthesis, Conformational Analysis, and Utilization in Medicinal Chemistry
Mr Luca GENTILUCCI
(UNIVERSITA DI BOLOGNA, Bologna, Italy)
12:35Lunch
Session Chair:
Prof. Yves FORT
(UNIVERSITÉ DE LORRAINE, Nancy, France)
14:00PL03 - The Importance of Heterocycles in Agrochemistry: Fungicides as a Case Study
Dr Harald WALTER
(SYNGENTA CROP PROTECTION AG BASEL, Basel, Switzerland)
14:55IL02 - Synthesis of Biorelevant Heterocycles with N-heterocyclic Carbenes
Prof. Andreas SCHMIDT
(TECHNICAL UNIVERSITY CLAUSTHAL, Clausthal-Zellerfeld, Germany)
15:25OC02 - Exploiting the Zincke Reaction to Produce Sophisticated Heptamethine Dyes
Dr Robert SMITH
(UNIVERSITY OF CENTRAL LANCASHIRE, Prestoin, United Kingdom)
15:40OC03 - Diverse Synthesis of Natural Product Inspired Fused and Spiro-Heterocyclic Scaffolds via Ring Distortion And Construction Strategy
Prof. Subhabrata SEN
(SHIV NADAR UNIVERSITY, Gautam Budh nagar, India)
15:55OC04 - Novel Cross-Conjugated Dienones Based on 4-Piperidone Moiety: Synthesis and Antitumor Properties
Dr Mikhail MAKAROV
(NESMEYANOV INSTITUTE OF ORGANOELEMENT COMPOUNDS OF RAS, Moscow, Russia)
16:10Coffee Break and Poster Session 1
18:00Welcome Reception (in the Exhibition area)
Tuesday June 9, 2015
Session Chair:
Dr Stéphanie HESSE
(UNIVERSITÉ DE LORRAINE, Metz, France)
09:00PL04 - Non Noble Metal Catalysis for Making Precious Molecules
Prof. Matthias BELLER
(UNIVERSITY OF ROSTOCK, Rostock, Germany)
09:55IL03 - Synthesis of Novel Alpha7-nAchR Ligands: from an Idea to in Rodent Results for Alzheimer [18F] TEP Imaging
Prof. Sylvain ROUTIER
(UNIVERSITÉ D'ORLÉANS, Orléans, France)
10:25OC05 - Recent Advances in the Total Synthesis of Phormidolides B and C
Mr Alejandro GIL ESCOLANO
(IRB BARCELONA, Barcelona, Spain)
10:40Coffee Break
Session Chair:
Prof. Patrick CHAIMBAULT
(UNIVERSITÉ DE LORRAINE, Metz, France)
11:10PL05 - Metal Catalysis for Heteroarene Synthesis
Prof. Michael GREANEY
(THE UNIVERSITY OF MANCHESTER, Manchester, United Kingdom)
12:05IL04 - New Methods in Thioamide Chemistry
Dr Mike PORTER
(UNIVERSITY COLLEGE LONDON, London, United Kingdom)
12:35Lunch
Session Chair:
Prof. Ferenc FULOP
(UNIVERSITY OF SZEGED, Szeged, Hungary)
14:00PL06 - The Discovery and Development of the HIV Intergrase Inhibitors Dolutegravir and Cabotegravir
Dr Brian JOHNS
(GLAXOSMITHKLINE, NC, United States)
14:55IL05 - Are Generic Drugs Only a Copy_and_Paste Products?
Prof. Stanislav RADL
(ZENTIVA, Prague, Czech Republic)
15:25OC06 - An Original Domino Radical Cyclisation/Smiles Rearrangement Combination: Application to the Synthesis of Indolo[2,3-b]Quinoline-Type Derivatives
Dr. Stéphane GERARD
(UNIVERSITÉ DE REIMS - CHAMPAGNE-ARDENNE, REIMS, France)
15:40OC07 - Palladium-Catalyzed Cross-Coupling Reactions in the Asymmetric Synthesis of Pyrrolo[1,2-b]Isoquinolines
Prof. Nuria SOTOMAYOR
(UNIVERSIDAD DEL PAÍS VASCO / EUSKAL HERRIKO UNIBERTSITATEA, Leioa - Bizkaia, Spain)
15:55OC08 - Synthesis of Long Regioregular Dialkyl-Substituted Alpha-Oligofurans
Dr Edward KORSHIN
(THE WEIZMANN INSTITUTE OF SCIENCE, Rehovot, Israel)
16:10Coffee Break and Poster Session 2
Wednesday June 10, 2015
Session chair:
Prof. John JOULE
(UNIVERSITY OF MANCHESTER, Manchester, United Kingdom)
09:00PL07 - Bronsted Acid and Metal-catalyzed Reactions in the Synthesis of Heterocycles
Prof. Esther LETE
(UNIVERSIDAD DEL PAÍS VASCO, Bilbao, Spain)
09:55IL06 - Utilization of Hypervalent Iodonium Reagents for the Construction and Functionalization of Heterocyclic Molecules
Dr Zoltan NOVAK
(EÖTVÖS UNIVERSITY, Budapest, Hungary)
10:25OC09 - Synthesis of Agrochemistry-Related F-Heterocycles from Novel Fluorinated Diazoalkanes
Dr Pavel MYKHAILIUK
(ENAMINE, Kyiv, Ukraine)
10:40Coffee Break
Session Chair:
Dr Harald WALTER
(SYNGENTA CROP PROTECTION AG BASEL, Basel, Switzerland)
11:15OC10 - Flavylium-Based Pigments – “Click” Synthesis & Biological Relevance
Dr Stefan CHASSAING
(ITAV, Toulouse, France)
11:30OC11 - Synthesis of 7-(2-Aminophenyl)- and 7-(4-Aminophenyl)Guanine, DNA Adducts Derived from the Phenylnitrenium Ion
Prof. Igor LINHART
(UNIVERSITY OF CHEMISTRY AND TECHNOLOGY, Prague, Czech Republic)
11:45OC12 - Heterocyclic Coumarine Analogs as Zinc Metalloprotease Inhibitors
Mr Peteris TRAPENCIERIS
(LATVIAN INSTITUTE OF ORGANIC SYNTHESIS, RIGA, Latvia)
12:00Lunch
Session chair:
Prof. Milan POTACEK
(MASARYK UNIVERSITY, Brno, Czech Republic)
13:30IL07 - Silicon-Containing Tetrahydrocyclopenta[C]Acridine Derivatives as CDKs Inhibitors: Design, Organometallic Synthesis, Metabolic Stability And Optimization
Prof. Philippe BELMONT
(UNIVERSITY PARIS DESCARTES, Paris, France)
14:00OC13 - Synthesis of Imidazo-Pyrrolo-Pyrazines/Diazepines/Diazocines via Domino Ugi/Micheal Reaction and Silver-Catalyzed Heteroannulation
Mr Zhenghua LI
(KU LEUVEN, Leuven, Belgium)
14:15OC14 - Synthesis and Antifungal Activity of N-Acyl Derivatives of 1,4-Benzoxazin- and 1,4-Benzoxazepin-3-ONES
Mrs Agata GOSZCZYNSKA
(WEST POMERANIAN UNIVERSITY OF TECHNOLOGY, SZCZECIN, Szczecin, Poland)
14:30OC15 - Mixed Cu(II) Cu(I) Complexes with Bioheterocycles as the Platform for Construction of Novel Anticancer Agents
Ms Olga KRASNOVSKAYA
(MOSCOW STATE UNIVERSITY, Moscow, Russia)
14:45Coffee Break
16:00Excursions
19:00Banquet
Thursday June 11, 2015
Session chair:
Prof. Henk VAN DER PLAS
(UNIVERSITY OF WAGENINGEN, Wageningen, The Netherlands)
09:00PL08 - Heterocycles Derived from Natural Products in Management of Multidrug Resistance
Prof. Ahcene BOUMENDJEL
(UNIVERSITÉ JOSEPH FOURIER, Grenoble, France)
09:55IL08 - At the Crossroads of Chemistry and Biology: Inhibiting Protein Kinase CK2 by Heterocyclic Small Molecules
Prof. Marc LE BORGNE
(UNIVERSITÉ CLAUDE BERNARD LYON 1, Lyon, France)
10:25Coffee Break
Session chair:
Prof. Jan BERGMAN
(KAROLINSKA INSTITUTE, Huddinge, Sweden)
11:00IL09 - Overcoming Resistance with beta-Lactams
Dr Eric DESARBRE
(BASILEA PHARMACEUTICA, Basel, Switzerland)
11:30OC16 - Discovery Of Novel Thieno[3,2-b]Pyrrole 5-Carboxamides as Potent Inhibitors of Chikungunya Virus (CHIKV)
Mr Kuan Chieh CHING
(NATIONAL UNIVERSITY OF SINGAPORE, Singapore, Singapore)
11:45Closing

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