EFMC-ASMC'15
Conferences > Archives > EFMC-ASMC'15
Sunday November 15, 2015
Session chair:
Prof. Hans Ulrich STILZ
(NOVO NORDISK, Malov, Denmark)
09:00Opening
Prof. Hans Ulrich STILZ (NOVO NORDISK, Malov, Denmark)
Prof. Koen AUGUSTYNS (UNIVERSITY OF ANTWERP, Antwerp, Belgium)
Dr Gene VAISBERG (CHEMBRIDGE CORPORATION, San Diego, United States)
Dr Raphael NUDELMAN (TEVA PHARMACEUTICAL INDUSTRIES, Petah Tikva, Israel)
09:30Directed Evolution of Stereoselective Enzymes: A Prolific Source of Catalysts for Asymmetric Reactions
Prof. Manfred T. REETZ
(MAX PLANCK INSTITUT FÜR KOHLENFORSCHUNG, Mulheim / Ruhr, Germany)
10:20Coffee break and Exhibition
10:50Studying and Targeting Deubiquitinases
Prof. Ashraf BRIK
(TECHNION-ISRAEL INSTITUTE OF TECHNOLOGY, Haifa, Israel)
11:35Setting a Course for Biomedical Innovation in the 21st Century
Dr Alan D. PALKOWITZ
(ELI LILLY & CO., Indianapolis, United States)
12:20Lunch and Exhibition
Session chair:
Dr Raphael NUDELMAN
(TEVA PHARMACEUTICAL INDUSTRIES, Petah Tikva, Israel)
14:00Traceless Transition Metal Catalysis for Synthetic Applications
Prof. Valentine P. ANANIKOV
(ZELINSKY INSTITUTE OF ORGANIC CHEMISTRY, Moscow, Russia)
14:45Protein Imprinted Polymers. What’s the Problem Here?
Dr Bernard S. GREEN
(SEMOREX TECHNOLOGIES, Ness Ziona, Israel)
15:30OC01 - A Synthetic and Predictive Approach to Unsymmetrical Biphenols by Iron-Catalyzed Chelated Radical-Anion Oxidative Coupling
Dr Doron PAPPO
(BEN-GURION UNIVERSITY, Beer Sheva, Israel)
15:45Coffee break and Exhibition
16:15OC02 - Development of Novel Nuclear Receptor Modulators Based on Silyl Functionality as Hydrophobic Core Structure
Dr Shinya FUJII
(UNIVERSITY OF TOKYO, Tokyo, Japan)
16:30Chemical Research in Space and under Microgravity Conditions
Dr Shimon AMSELEM
(SPACEPHARMA, Herzliya Pituach, Israel)
17:15Targeted Cancer Diagnosis and Therapy with Peptide Conjugates
Prof. Annette BECK-SICKINGER
(LEIPZIG UNIVERSITY, Leipzig, Germany)
18:00Closing of the day
19:30Welcome Reception
Monday November 16, 2015
Session chair:
Dr Gene VAISBERG
(CHEMBRIDGE CORPORATION, San Diego, United States)
08:30Crystalline Sponge Method as Applied to Pharmaceutical Studies
Prof. Makoto FUJITA
(UNIVERSITY OF TOKYO, Tokyo, Japan)
09:15Stimuli-Responsive Drug Carriers for Controlled Delivery and Nano-Medicine Applications
Prof. Itamar WILLNER
(THE HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel)
10:05Coffee break and Exhibition
10:35Quinone-Methide Species - a Gateway to Functional Molecular Systems
Prof. Doron SHABAT
(TEL AVIV UNIVERSITY, Tel Aviv, Israel)
11:20Exploration of Innovative Chemical Space for Biological Screening: the European Lead Factory Perspective
Dr Fabrizio GIORDANETTO
(TAROS CHEMICALS, New York, United States)
12:05OC04 - Hypervalent Iodine Fluoroalkylating Reagents - Going Beyond Trifluoromethylation
Ms Julie CHARPENTIER
(ETH ZÜRICH, Zürich, Switzerland)
12:20Lunch and Exhibition
Poster SessionCompany Workshops
13:00Poster session (even numbers)
13:00Moving from Small Molecule Patent Searching to Patent Evaluation - Applications of SciFinder with PatentPak
Mr Paul PETERS
(CAS, Hannover, Germany)
Session chair:
Dr Doron PAPPO
(BEN-GURION UNIVERSITY, Beer Sheva, Israel)
14:00The Art of Building Small
Prof. Ben FERINGA
(UNIVERSITY OF GRONINGEN, Groningen, The Netherlands)
14:45Personalized Medicine - Will it Really Happen?
Dr Aharon SCHWARTZ
(SCHWARTZ INNOVATIONS, Mevaseret Zion, Israel)
15:30OC05 - Multi-Responsive Polymeric Assemblies
Dr Roey AMIR
(SCHOOL OF CHEMISTRY - TEL AVIV UNIVERSITY, Tel Aviv, Israel)
15:45Coffee break and Exhibition
16:15Expanding Medicinal Chemistry Space: The Compact Module Initiative and Beyond
Dr Jean-Marc PLANCHER
(F. HOFFMANN-LA ROCHE, Basel, Switzerland)
17:00Assembly Line Synthesis
Prof. Varinder K. AGGARWAL
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom)
17:45Closing of the day
Tuesday November 17, 2015
Session chair:
Prof. Koen AUGUSTYNS
(UNIVERSITY OF ANTWERP, Antwerp, Belgium)
08:30Harnessing Fluorine - Induced Ion - Dipole Attractive Forces in Enantioselective Catalysis
Prof. Amir H. HOVEYDA
(BOSTON COLLEGE, Chestnut Hill, United States)
09:15Drug Discovery in the Ubiquitin Pathway : the E3 Ligases
Dr Philippe NAKACHE
(METABOMED, Yavne, Israel)
10:00OC06 - Computational Discovery of Liposomal Drugs: from in Silico Predictions to in Vivo Validation
Prof. Amiram GOLDBLUM
(HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel)
10:15Coffee break and Exhibition
10:45Tailor-made Enzymes –Nature’s and Ours
Dr Dan TAWFIK
(WEIZMANN INSTITUTE OF SCIENCE, Rehovot, Israel)
11:30Discovery of a Potent and Selective Reversible BTK Inhibitor for the Treatment of Autoimmune Diseases
Dr Robert PULZ
(NOVARTIS PHARMA, Basel, Switzerland)
12:15Prize Ceremony
12:20EFMC Prize for a Young Medicinal Chemist in Academia
Achieving Intra-BET Selectivity of BET Bromodomain Chemical Probes: Bump-And Hole and PROTAC Approaches
Prof. Alessio CIULLI
(UNIVERSITY OF DUNDEE, Dundee, United Kingdom)
12:35EFMC Prize for a Young Medicinal Chemist in Industry
Structure-Based Drug Design with G Protein-Coupled Receptors
Dr Steve ANDREWS
(HEPTARES, Welwyn Garden City, United Kingdom)
12:50Lunch and Exhibition
Poster SessionCompany Workshops
13:15Poster Session (odd numbers)
13:15Data-Driven Approaches to Medicinal Chemistry
Mr Joannis TELIORIDIS
(ELSEVIER, Amsterdam, The Netherlands)
14:15Free afternoon
15:00Excursions
Wednesday November 18, 2015
Session chair:
Dr Micha FRIDMAN
(TEL AVIV UNIVERSITY, Ramat Aviv, Tel Aviv, Israel)
08:30Versatile Iridium Catalysts for a Broad Range of Asymmetric Transformations
Prof. Erick M. CARREIRA
(ETH ZÜRICH, Zürich, Switzerland)
09:20Challenges and Synthetic Ingenuity in the Generic World
Dr Lilach HEDVATI
(TEVA, Petah-Tiqva, Israel)
10:00OC07 - Synthesis and Application of Unnatural Proline Analogues: Advanced Building Blocks for Medicinal Chemistry
Dr Pavel MYKHAILIUK
(ENAMINE, Kyiv, Ukraine)
10:15Coffee break and Exhibition
10:45Evolving GPCRs to Favorable Biophysical Properties: Enabling Drug Screening and Structural Studies
Prof. Andreas PLÜCKTHUN
(UNIVERSITY OF ZÜRICH, Zurich, Switzerland)
11:35The Power of Integrated Technological Platforms to Advance Science and Medicine
Dr Berta STRULOVICI
(WEIZMANN INSTITUTE OF SCIENCE, Rehovot, Israel)
12:15OC08 - Necrosis: Cellular Mechanisms and Treatment
Prof. Amnon ALBECK
(BAR ILAN UNIVERSITY, Ramat Gan, Israel)
12:45Lunch and Exhibition
Session chair:
Prof. Ilan MAREK
(ISRAEL INSTITUTE OF TECHNOLOGY, Haifa, Israel)
14:00OC09 - Catalytic Asymmetric Synthesis of Caprazamycin B and Caprazol
Dr Takumi WATANABE
(INSTITUTE OF MICROBIAL CHEMISTRY (BIKAKEN), Tokyo, Japan)
14:15OC10 - Synthesis of Archazolid F and Other Novel Archazolids: Highly Potent V-Atpase Inhibitors
Mr Stephan SCHEEFF
(UNIVERSITY OF BONN, Bonn, Germany)
14:30OC11 - Protecting Group-Free Strategies for The Synthesis of Nucleosides
Mr Mike DOWNEY
(INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY, Prague-6, Czech Republic)
14:45OC12 - Development of Anti-Influenza Drugs
Prof. Jim-Min FANG
(NATIONAL TAIWAN UNIVERSITY, Taipei, Taiwan)
15:00OC13 - Cross Metathesis of Sulfonamides and Sulfoxides
Mr Adam RAJKIEWICZ
(UNIVERSITY OF WARSAW, Warsaw, Poland)
15:15Coffee break and Exhibition
15:45The Barry Cohen Award for Excellence in Medicinal Chemistry Prize Ceremony
Synthesis-Informed Design Directed at Transformative Therapies: Eradication of Hiv/Aids, Alzheimer's Disease and Resistant Cancer
Prof. Paul A. WENDER
(STANFORD UNIVERSITY, Stanford, United States)
16:30Closing remarks
Prof. Ilan MAREK
(ISRAEL INSTITUTE OF TECHNOLOGY, Haifa, Israel)
20:00Banquet

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