EFMC-YMCS 2019
Conferences > Archives > EFMC-YMCS 2019
Thursday 05/09/2019
14:15Registration
15:00Welcome and Opening
Session Chair:
Prof. Emmanouil FOUSTERIS
(UNIVERSITY OF PATRAS, Patras, Greece)
15:05KL01 - The Emergence of Antibody-Drug Conjugates (ADCs) as Targeted Cancer Therapies: From Ehrlich's "Magic Bullet" Concept to Calicheamicin γ1I and Mylotarg
Prof. K.C. NICOLAOU
(RICE UNIVERSITY, Houston, United States)
EFMC-YMCS Competition Presentation Session I
15:35OC01 - Functionalization of Tumour-Targeting Antibodies Via Enzymatic Oxidation of Tyrosine to 1,2-Quinones
Winner of the Young Medicinal Chemist Meeting in The Netherlands
Mr Jorick BRUINS
(WAGENINGEN UNIVERSITY, WAGENINGEN, The Netherlands)
15:55OC02 - Synthetic Small Molecules Interfering with Oncogenic Micrornas for the Induction of Glioblastoma Stem Cells Differentiation
Winner of the Young Medicinal Chemist Meeting in France
Dr Chloé MAUCORT
(INSTITUTE OF CHEMISTRY OF NICE, Val de Reuil, France)
16:15OC03 -New Ruthenium-Cyclopentadienyl Complexes Bearing Biotinylated (Macro)Ligands: Targeting Strategies to Fight Metastatic Breast Cancer
Winner of the Young Medicinal Chemist Meeting in Portugal
Dr Leonor CORTE-REAL
(CENTRO DE QUÍMICA ESTRUTURAL, Lisboa, Portugal)
16:35Flash Poster Presentations (01-10)
FP01 - A New Life for Diazaborines: the Next Generation of Serine Protease Inhibitors
Mr Joao ANTONIO
(UNIVERSITY OF LISBON, Lisbon, Portugal)
FP02 - From Peptides to Peptidomimetics: Structure-Activity Relationship of a Factor H-Binding Peptide to Modulate Undesired Host Complement Activity
Dr Clément BECHTLER
(UNIVERSITY OF BASEL, Wuppertal, Germany)
FP03 - Matrix Metalloproteinase-12 Inhibitors: Synthesis, Structure-Activity Relationships and Intestinal Absorption of Novel Sugar-Based Biphenylsulfonamide Carboxylates
Dr Doretta CUFFARO
(UNIVERSITY OF PISA, Pisa, Italy)
FP04 - Photophysical Properties and Antiparasitic Activity of Bodipy-Tethered Dinuclear Trithiolato-Bridged Ruthenium(II)-Arene Complexes
Mrs Oksana DESIATKINA
(UNIVERSITY OF BERN, Bern, Switzerland)
FP05 - N-ALKYL L-Iminosugars as Novel Anti-Inflammatory and Anti-Biofilm Tools for Cystic Fibrosis Lung Infections
Ms Anna ESPOSITO
(UNIVERSITY OF NAPOLI FEDERICO II, Napoli, Italy)
FP06 - Design, Synthesis and Biological Evaluation of Novel Substituted Purine Isosters as EGFR Kinase Inhibitors, with Promising Pharmacokinetic Profile and In Vivo Efficacy
Dr Efthymios-Spyridon GAVRIIL
(NATIONAL AND KAPODISTRIAN UNIVERSITY OF ATHENS, Athens, Greece)
FP07 - Metal-Chelating Acetohydroxamic Acids Against Hepatitis C Virus and Flaviviruses
Ms Erofili GIANNAKOPOULOU
(NATIONAL AND KAPODISTRIAN UNIVERSITY OF ATHENS, Athens, Greece)
FP08 - Discovery of Small-Molecule Modulators of 14-3-3 PPIs Via Dynamic Combinatorial Chemistry
Mr Alwin HARTMAN
(UNIVERSITY OF GRONINGEN, Groningen, The Netherlands)
FP09 - Purine Nucleoside Analogs as Highly Potent Leads for the Treatment of Human African Trypanosomiasis
Dr Fabian HULPIA
(UGENT, Beerse, Belgium)
FP10 - Development of Allosteric Inhibitors of ColH Using DCC Strategy
Dr Jelena KONSTANTINOVIC
(HELMHOLTZ INSTITUTE FOR PHARMACEUTICAL RESEARCH SAARLAND (HIPS), Saarbrücken, Germany)
16:55Coffee Break
EFMC-YMCS Competition Presentation Session II
Session Chair:
Dr Kristina GONCHARENKO
(SPIROCHEM AG, Basel, Switzerland)
17:10OC04 - Novel Acridine Derivatives as TDP 1 and/or 2 Inhibitors
Winner of the Young Medicinal Chemist Meeting in Greece
Mrs Maria KARELOU
(NATIONAL AND KAPODISTRIAN UNIVERSITY OF ATHENS, Athens, Greece)
17:30OC05 - Discovery of a Novel Chemotype of Non-Acidic, Neutral and Macrocyclic Keap1 Inhibitors
Winner of the Young Medicinal Chemist Meeting in Sweden
Mr Fabio BEGNINI
(UPPSALA UNIVERSITY, Uppsala, Sweden)
17:50OC06 - Directed Evolution of Short Peptides for Selective Detoxification of Lead
Winner of the Young Medicinal Chemist Meeting in Switzerland
Dr Michal SHOSHAN
(UNIVERSITY OF ZURICH, Zürich, Switzerland)
18:10Flash Poster Presentations (11-20)
FP11 - Identification, Synthesis and Optimization of Inhibitors of the Protein Tyrosine Phosphatase SHP2
Dr Yelena MOSTINSKI
(LEIBNIZ-FORSCHUNGSINSTITUT FÜR MOLEKULARE PHARMAKOLOGIE, Rishon LeZion, Israel)
FP12 - Multitarget Triazoles: an Innovative Approach for the Treatment of Alzheimer’s Disease
Ms Vanesa NOZAL GARCIA
(CIB - CSIC, Madrid, Spain)
FP13 - TDP-43 Modulation by CDC7 Inhibitors as a Therapeutic Strategy for Amyotrophic Lateral Sclerosis
Ms Elisa ROJAS
(CIB - CSIC, Madrid, Spain)
FP14 - Use of the 4-Hydroxy-Triazole Moiety as a Bioisosteric Tool in the Development of Selective Ligands for Subtypes Ampa Receptor
Dr Stefano SAINAS
(UNIVERSITY OF TORINO, Torino, Italy)
FP15 - In Vitro and In Ovo Evaluation of Ros-Activatable Anticancer Boronate Prodrugs of Doxorubicin
Dr Charles SKARBEK
(UNIVERSITY PARIS SUD, Orsay, France)
FP16 - Design and Synthesis of Tead's Ligands for the Treatment of Cancers
Mrs Manon STURBAUT
(UNIVERSITY OF LILLE, Lille, France)
FP17 - Drug-Fragment Based Explorations for Novel Enterovirus Inhibitors
Ms Clara VAN HOEY
(UNIVERSITY OF VIENNA, Vienna, Austria)
FP18 - Gemcitabine-GnRH Bioconjugates Bearing Oxime Bond Linkages: Synthesis, In Vitro Stability, Drug Release and Cytotoxic Effect
Dr Eirinaios VRETTOS
(UNIVERSITY OF IOANNINA, Ioannina, Greece)
FP19 - Development of GSTO1-1 Inhibitors for the Treatment of Inflammatory Conditions
Ms Yiyue XIE
(MONASH UNIVERSITY, Melbourne, Australia)
FP20 - Identification of a Novel Quinoline-Based DNA Demethylating Compound Highly Potent in Cancer Cells
Dr Clemens ZWERGEL
(UNIVERSITY OF ROME LA SAPIENZA, Rome, Italy)
18:30EFMC-YMCS Poster Presentation Session 1 (Odd), Bites & Drinks
19:30EFMC-YMCS Poster Presentation Session 2 (Even), Bites & Drinks
20:30End of the Scientifc Programme
EFMC-YSN Soft Skills Training Session (1)
20:30How to Boost Your Oral Presentation Skill, and Create a Good Slideshow
Dr Kristina GONCHARENKO
(SPIROCHEM AG, Basel, Switzerland)
20:45Getting the Job You Deserve!
Dr. David ALKER
(DAVID ALKER ASSOCIATES, Birchington, United Kingdom)
21:15EFMC-YSN Networking Event
22:30End of the Day
Friday 06/09/2019
08:29EFMC-YMCS Competition Presentation Session III
Session Chair:
Dr Cassandra LEE FLEMING
(UNIVERSITY OF GOTHENBURG, Gothenburg, Sweden)
08:30KL02 - Medicinal Chemistry Between Serendipity and (Artificial) Intelligence
Dr Cornelia ZUMBRUNN
(IDORSIA PHARMACEUTICALS, Allschwil, Switzerland)
09:00OC07 - Antiplasmodial Activity of SAHAquines, Novel SAHA - Primaquine Hybrids
Winner of the Young Medicinal Chemist Meeting in Croatia
Dr Maja BEUS
(UNIVERSITY OF ZAGREB, Zagreb, Croatia)
09:20OC08 - Hybrdization Approach Towards Novel Antituberculars: Design, Synthesis, And Antimicrobial Evaluation Hybrid Compounds Combining Pyrazinamide and p Aminosalicylic Acid
Winner of the Young Medicinal Chemist Meeting in Czech Republic
Dr Ghada BOUZ
(CHARLES UNIVERSITY, Hradec Kralove, Czech Republic)
09:40OC09 - Synthesis, Computational and Biological Evaluation of Novel Benzimidazole Compounds for the Treatment of Cryptococcus Neoformans
Winner of the Young Medicinal Chemist Meeting in the United Kingdom
Ms Gina WASHBOURN
(UNIVERSITY OF LIVERPOOL, Liverpool, United Kingdom)
10:00OC10 - Nʼ-Benzylated Derivatives of N-(7-Chloroquinolin-4-Yl)Octane-1,8-Diamine as Quorum Sensing Inhibitors in Pseudomonas Aeruginosa
Winner of the Young Medicinal Chemist Meeting in Serbia
Ms Marta SPASIC
(UNIVERSITY OF BELGRADE, Nis, Serbia)
10:20Coffee Break
EFMC-YMCS Competition Presentation Session IV
Session Chair:
Dr Eleni PONTIKI
(ARISTOTELE UNIVERSITY OF THESSALONIKI, Thessaloniki, Greece)
10:40OC11 - Geometric Isomers of N-Propargyl-4-Syrylpiperidine Discriminate Between Monoamine Oxidase Isoforms A and B
Winner of the Young Medicinal Chemist Meeting in Slovenia
Dr Damijan KNEZ
(UNIVERSITY OF LJUBLJANA, Ljubljana, Slovenia)
11:00OC12 A Fusing Strategy Application: Towards Potent ChE Inhibitors With MTDL Profile
Winner of the Young Medicinal Chemist Meeting in Turkey
Dr Gülsah BAYRAKTAR
(EGE UNIVERSITY FACULTY OF PHARMACY, Izmir, Turkey)
11:20OC13 - Development of Unique Molecular Probes: Low-Basicity Agonists for the Study of 5-HT7 Receptor Function
Winner of the Young Medicinal Chemist Meeting in Poland
Dr Adam HOGENDORF
(MAJ INSTITUTE OF PHARMACOLOGY, POLISH ACADEMY OF SCIENCES, Krakow, Poland)
11:40OC14 - The Establishment of Tocopherol Reference Intervals for Hungarian Adult Population Using Validated HPLC Method
Winner of the Young Medicinal Chemist Meeting in Hungary
Dr Gábor VERES
(HUNGARIAN ACADEMY OF SCIENCES, Budapest, Hungary)
12:00Lunch
EFMC-YSN Soft Skills Training Session (2)
13:00Why Was My Paper Rejected? Tips from an Editor on How to Get Published
Dr David PERALTA
(WILEY-VCH VERLAG GMBH & CO. KGAA, Weinheim, Germany)
EFMC-YMCS Competition Presentation Session V
13:45Session Chair:
Prof. Grigorios ZOIDIS
(UNIVERSITY OF ATHENS, Athens, Greece)
13:45OC15 - Expanding the Chemical Space of DNA-Encoded Small Molecule Libraries
Winner of the Young Medicinal Chemist Meeting in Germany
Dr Andreas BRUNSCHWEIGER
(TU DORTMUND, Dortmund, Germany)
14:05OC16 - Finding the Right Candidate for the Right Position: a Fast NMR-Assisted Combinatorial Method for Optimizing Nucleic Acids Binders
Winner of the Young Medicinal Chemist Meeting in Spain
Dr Andrés GONZALEZ SANTANA
(IQOG - CSIC, Madrid, Spain)
14:25OC17 - From ZINC to ZINClick: Our Way to Explore the Chemical Space
Winner of the Young Medicinal Chemist Meeting in Italy
Prof. Alberto MASSAROTTI
(UNIVERSITY OF EASTERN PIEDMONT, Novara, Italy)
14:45OC18 - Extended Glucuronides: Achieving Site-Selectivity Through Extracellular Drug Release
Winner of the Young Medicinal Chemist Meeting in Denmark
Mr Raoul WALTHER
(AARHUS UNIVERSITY, Aarhus, Denmark)
15:05OC19 - Cyclopropenium-Based Polymers
Winner of the Young Medicinal Chemist Meeting in Israel
Mr Noam STEINMAN
(HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel)
15:25Voting Break
15:40KL03 - Chemical Tools to Target and Image Tumours
Prof. Stuart CONWAY (UNIVERSITY OF OXFORD, Oxford, United Kingdom)
 (BIOIBÉRICA)
16:10Closing and Award Ceremony
16:20End of the Symposium

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