EFMC-ISMC 2016

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EFMC Best Poster Prizes

The EFMC Best Poster Prizes have been granted to the following participants :

  • P096 - Yasuhiro Imaeda (Takeda Pharmaceutical Company, Japan)
    DISCOVERY OF TAK-272: A NOVEL, POTENT AND ORALLY ACTIVE RENIN INHIBITOR

  • P036 - Dmitrii Kalinin (University of Münster, Germany)
    DESIGN, SYNTHESIS AND ANTIBACTERIAL ACTIVITY OF PROLINE HYDROXAMATES TARGETING ZINC-DEPENDENT ENZYMES

  • P132 - Nis Halland (Sanofi, Germany)
    NOVEL SMALL MOLECULE INHIBITORS OF ACTIVATED THROMBIN ACTIVATABLE FIBRINOLYSIS INHIBITOR (TAFIa) FROM NATURAL PRODUCT ANABAENOPEPTIN

  • P192 - Geoffrey Schwertz (ETH Zurich, Switzerland)
    SHMT INHIBITION: A NEW HOPE TO DEFEAT MALARIA

  • P253 - Xavier Lucas (University of Dundee, United Kingdom)
    PROTACTING LEADS: DESIGN OF A PROTEIN SURFACE-TARGETING FRAGMENT LIBRARY

  • P334 - Jonas Kaindl (Friedrich-Alexander-University Erlangen-Nuernberg, Germany)
    STRUCTURE-GUIDED DEVELOPMENT AND MOLECULAR MODELLING OF D2R/NTS1R HETERODIMER-SELECTIVE LIGANDS

  • P444 - Arno Vermote (Ghent University, Belgium)
    POTENTIATOR DRUGS FOR BAD BUGS - HAMAMELITANNIN ANALOGUES POTENTIATE ANTIBIOTICS IN THE FIGHT AGAINST STAPHYLOCOCCUS AUREUS

  • P466 - Liam Hudson (Institute of Cancer Research, United Kingdom)
    DEVELOPMENT OF A NEW CLASS OF ALK2 INHIBITOR FOR THE STUDY OF THE MOST AGGRESSIVE PAEDIATRIC BRAIN CANCER, DIPG

  • P592 - Christian Kersten (Johannes Gutenberg University, Germany)
    SELECTIVITY DETERMINING FEATURES IN N-MYRISTOYLTRANSFERASES - A POTENTIAL DRUG TARGET WITH A HIGHLY CONSERVED BINDING SITE

  • P522 - Daniela Dengler (Friedrich-Alexander University Erlangen-Nuremberg, Germany)
    DISCOVERY OF A G-PROTEIN BIASED MU OPIOID ANALGESIC WITH REDUCED SIDE EFFECTS

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