Small Becomes Big in Medicinal Chemistry: Fragment-based Drug Discovery
Oegstgeest (near Leiden), The Netherlands April 28-May 1, 2019
Registration
Dinner
Breakfast
Opening
Introduction to Fragment Based Discovery – Overview of the Process and a Historical Perspective
Coffee Break
Design Principles for Fragment Libraries
Lunch
Experiences and Issues with Biochemical Assays in Fragment-Based Drug Discovery
Coffee Break
Day End
Walking tour through Leiden
Dinner in Leiden
Breakfast
Why Fragments Make Sense and Actually Work
Coffee Break
Computational Approaches for Fragment Screening and Fragment Evolution
Lunch
Coffee Break
Application-Project in group (Part 1)
Day End
Dinner
Breakfast
Application-Project in group (Part 2)
Coffee Break
Presentations of the results
Wrap-up and Lunch