A Matter of Time: A Kinetic Perspective on Drug-Target Interactions
Oegstgeest (near Leiden), The Netherlands April 23-26, 2017
Registration
Dinner
Breakfast
Introduction
Coffee Break
Lunch
Characterizing the Dynamics of Molecular Interactions
Prof. Helena DANIELSON
UPPSALA UNIVERSITY, Uppsala, Sweden
Coffee Break
Characterizing the Dynamics of Molecular Interactions - Part II
Prof. Helena DANIELSON
UPPSALA UNIVERSITY, Uppsala, Sweden
Day End
Dinner and walking tour through Leiden
Breakfast
Kinetics for drug discovery: In vitro assays to study GPCRs
Dr Laura HEITMAN
UNIVERSITY OF LEIDEN, Leiden, The Netherlands
Coffee Break
Kinetics in Drug Discovery - A Case for G Protein-coupled Receptors
Prof. Ad P. IJZERMAN
UNIVERSITY OF LEIDEN, Leiden, The Netherlands
Lunch
Pharmacokinetic-pharmacodynamic Relationships, the Connecting Role of Binding Kinetics
Dr Liesbeth DE LANGE
UNIVERSITY OF LEIDEN, Leiden, The Netherlands
Coffee Break
Pharmacokinetic-pharmacodynamic Relationships, the Connecting Role of Binding Kinetics - Part II
Mr Wilbert DE WITTE
UNIVERSITY OF LEIDEN, Leiden, The Netherlands
Day End
Dinner
Breakfast
The Use of Kinetic Data in Early Drug Discovery: HSP90 as a Model to Gain Mechanistic Insight into Drug Binding Kinetics
Dr Matthias FRECH
MERCK, Darmstadt, Germany
Coffee Break
The Use of Kinetic Data in Early Drug Discovery: HSP90 as a Model to Gain Mechanistic Insight into Drug Binding Kinetics - Part II
Dr Matthias FRECH
MERCK, Darmstadt, Germany
Wrap-up and Lunch