A Matter of Time: A Kinetic Perspective on Drug-Target Interactions
Oegstgeest (near Leiden), The Netherlands April 23-26, 2017
Registration
Dinner
Breakfast
Introduction
Coffee Break
Lunch
Characterizing the Dynamics of Molecular Interactions
Coffee Break
Characterizing the Dynamics of Molecular Interactions - Part II
Day End
Dinner and walking tour through Leiden
Breakfast
Kinetics for drug discovery: In vitro assays to study GPCRs
Coffee Break
Kinetics in Drug Discovery - A Case for G Protein-coupled Receptors
Lunch
Pharmacokinetic-pharmacodynamic Relationships, the Connecting Role of Binding Kinetics
Coffee Break
Pharmacokinetic-pharmacodynamic Relationships, the Connecting Role of Binding Kinetics - Part II
Day End
Dinner
Breakfast
The Use of Kinetic Data in Early Drug Discovery: HSP90 as a Model to Gain Mechanistic Insight into Drug Binding Kinetics
Coffee Break
The Use of Kinetic Data in Early Drug Discovery: HSP90 as a Model to Gain Mechanistic Insight into Drug Binding Kinetics - Part II
Wrap-up and Lunch