ECHC 2016

XXVII European Colloquium on Heterocyclic Chemistry

 Amsterdam, The Netherlands    July 3-6, 2016

Opening Lecturer

Prof. Herbert WALDMANN
Opening Lecture - PL01 - How Natural Products Can Inspire Chemical Biology and Drug Discovery
 
 

Plenary Lecturers

Prof. Martin D. BURKE
PL06 - Making Molecular Prosthetics with a Small Molecule Synthesizer
Prof. Dieter ENDERS
PL02 - Organocatalytic Asymmetric Synthesis of Heterocycles
Prof. Karl Anker JOERGENSEN
PL07 - Organocatalysis for Diversity-Oriented Synthesis
Dr Fernando LOPEZ
PL04 - Carbo- and Heterocycles via Metal-Catalyzed Cycloadditions
Prof. Floris RUTJES
PL03 - Catalytic Approaches from the Synthesis of Enantiopure Biologically Relevant Heterocycles
Prof. Jerome WASER
PL05 - Springer Junior Heterocyclic Chemistry Award Lecture (chaired by Bert Maes, editor of Springer)
Exploiting the Reactivity of Strained Rings and Hypervalent Bonds for the Synthesis of Heterocycles

Invited Lecturers

Prof. Lutz ACKERMANN
IL10 - C-H Functionalization for the Synthesis and Assembly of Heterocycles
Prof. Luca BANFI
IL03 - Stereoselective Heterocycle Synthesis Coupling Multicomponent Reactions with Biocatalysis or Organocatalysis
Prof. Geert-Jan BOONS
IL04 - Metal Free Cllick Reactions For Glycoconjugate Modification
Prof. Iain COLDHAM
IL13 - Metallation–Substitution of Saturated Nitrogen Heterocycles
Prof. Gwilherm EVANO
IL06 - Ynamides: Remarkable Building Blocks for Heterocyclic Synthesis
Prof. Gianluca M. FARINOLA
IL07 - Photoactive Molecular and Supramolecular Materials Built-up with Heterocycles
Prof. Karl GADEMANN
IL08 - Redesigning the Molecules of Nature: Lessons Learned from Total Synthesis
Prof. Syuzanna HARUTYUNYAN
IL09 - Copper Catalysis for Synthesis of Enantiopure Alcohols, Amines and Heteroarenes
Prof. Laurence HARWOOD
IL02 - The Development of Ligand Systems for Separating Minor Actinides from Lanthanides for Nuclear Fuel Reprocessing
Prof. Xiaoguang LEI
IL12 - Complex Natural Product as a Driving Force for Discovery in Organic Synthesis and Chemical Biology
Dr Geraldine MASSON
IL11 - Catalysis: A Versatile Tool for the Synthesis of Nitrogen-Containing Heterocycles
Dr Gerhard MÜLLER
IL05 - Target Family-Centric Privileged Structures: a Rich Playground for Diverse Heterocyclic Chemotypes
Prof. Dr Valentine G. NENAJDENKO
IL14 - α-Perluoroalkylated Cyclic Imines as a Valuable Building Blocks
Prof. Thomas NIELSEN
IL15 - New Strategies for the Synthesis of Heterocyclic through Multicomponent Reactions and Metal-Catalyzed Isomerization
Prof. Tobias RITTER
IL01 - Fluorinated Imaging Materials

Keynote Lecture

Dr Laurent COMMEIRAS
KL07 - Gamma-Alkylidenebutenolides and Gamma-Hydroxybutyrolactams: Preparation and Reactivity
Dr Daniel GARCÍA RIVERA
KL06 - New Multicomponent Reactions and Strategies to Heterocyclic and Macrocyclic Peptides
Prof. Christopher HULME
KL02 - First-in-Class MCRs Coupled with Cascade Reactions for the Generation of Molecular Complexity
Prof. Norbert KRAUSE
KL05 - Synthesis of New Spiroacetals by Sustainable Gold Catalysis
Dr Andrew LAWRENCE
KL03 - Biomimetic Natural Product Synthesis
Dr Timothy NOEL
KL08 - Functionalization of Heterocycles via C–H Activation and Photoredox Catalysis in Batch and Continuous Flow
Prof. Till OPATZ
KL01 - Alpha-Functionalization of Amines as a Tool for the Synthesis of Heterocycles and Natural Products
Dr Sven RUF
KL09 - Going Beyond ß-Amino Acid Derivatives as Inhibitors of Cathepsin A
Prof. Johan WINNE
KL04 - New Tricks for Old Heterocycles: from Natural Product Synthesis to Click-Like Functionalizations

Oral Communication

OC19 - Pd- and Cu-Catalyzed Stereo- and Regiocontrolled Decarboxylative / C-H Alkenylation of Heroarenes
Ms Emma BLACKHAM
OC08 - Combining Photochemistry and Catalysis: Rapid Access to SP3 - Rich Polyheterocycles from Simple Pyrroles
Mr John BRAUN
OC09 - Intramolecular Tsuji-Trost Cascade Cyclization as a Novel Synthetic Strategy Towards Muironolide A
Mr Timothée CADART
OC20 - Enantioselective Organocatalyzed Α-Sulfanylation of Isoxazolidin-5-ones: An Approach To b2,2-Amino Acids
Ms Rekha CHADDA
OC13 - The Allylic Azide Rearrangement in Tandem with Huisgen Cycloaddition: Synthesis of Diverse Polyhydroxylated Nitrogen Containing Scaffolds
Mr Giacomo CRISENZA
OC17 - Brönsted-Acid Catalysed C2-Alkenylation of Aromatic Nitrogen Heterocycles
Dr Doris DALLINGER
OC40 - A Lab-Scale Reactor for the Continuous Generation of Anhydrous Diazomethane
Prof. Roman DEMBINSKI
OC05 - Synthesis of Highly and Diversely Substituted Heterocycles from Alk-3-yn-1-ones (Propargyl Ketones)
Mr Mohamed EL GHOZLANI
OC14 - Synthesis and Potential Cytotoxic Activity of New Substituted Indazole Derivatives Bearing Pyrrole and 2-Pyrone
Dr Martin FEITERS
OC36 - N-Heterocyclic Carbene Ligands in Iridium Complexes for the Detection of Pyridine Analogues in NMR by Non-Hydrogenative Para-Hydrogen Induced Hyperpolarization
Dr M. Angeles FERNANDEZ-IBANEZ
OC31 - Picolinic Acid Ligand-Promoted Palladium-Catalyzed C-H Acetoxylation of Simple Arenes
Mr Christian FISCHER
OC38 - Direct Heteroatom Incorporating Ester to Arene Transformation: Modular Synthesis of Fluorescent Dyes
Mr Fernando FUMAGALLI
OC02 - Efficient Approach to the Synthesis of 2,3-Substituted Furo[2,3-b]Pyridines
Ms Larissa GEIGER
OC33 - Scope and Limitations of the Organocatalyzed Domino Vinylogous Aldol Oxa Michael Reaction
Mr Andrea GINI
OC07 - Synthesis of 3-Benzazepines by Metal-Free Oxidative C-H Bond Functionalization-Ring Expansion Tandem Reaction
Dr Agnieszka GRAJEWSKA
OC43 - Novel Synthesis of Tetrahydroisoquinoline Derivatives Using Petasis Reaction
Dr Michael HALL
OC25 - Chirality in Boron-Chelated Dipyrromethene Fluorophores: Synthesis and Chiroptical Investigations
Mr Mickel HANSEN
OC42 - Photopharmacology
Mr Josh HOMER
OC15 - Towards a Biomimetic Synthesis of Sciodole
Prof. Yoichi HOSHIMOTO
OC01 - Poxim: A Novel N-Heterocyclic Carbene Equipped with Multifunctional Phosphine Oxide
Dr Steen INGEMANN JORGENSEN
OC06 - Asymmetric Synthesis of Natural Tetrahydroisoquinolines and Tetrahydroprotoberberines
Mr Art KRUITHOF
OC35 - Integrative Methodology for Iterative Theory-Experiment Driven Multicomponent Reaction Development
Mr Petrus KUIJPERS
OC22 - Aliphatic N-Heterocycle Synthesis through Direct C-H Bond Amination
Prof. Tibor KURTÁN
OC32 - Stereoselective Transformations of 2h-Chromene Derivatives
Dr Julien LOUVEL
OC41 - Designing Residence Time into Heterocyclic Ligands for Drug Targets
Mr Josep MAS ROSELLO
OC44 - Palladium Catalyzed C-Arylation of Amino Acid Derived Hydantoins
Dr Matthew MCLACHLAN
OC12 - Exploring Tryptophan Synthase as a Herbicidal Mode of Action
Prof. José Carlos MENÉNDEZ
OC29 - Biology-Oriented Synthesis Based on Privileged Structures: Building Framework Diversity Around Pyrrole Cores
Mrs Solène MIASKIEWICZ
OC21 - Is Gold Catalysis a Competitive Method toward Heterocycles ?
Prof. Abraham NUDELMAN
OC27 - Biologically Active Indolines - Novel Multi-Functional Indolinic Drugs for the Treatment of Inflammatory Diseases
Ms Ophélie QUINONERO
OC45 - Enantioselective Synthesis of 4-Arylpyridine Atropisomers by Central-to-Axial Chirality Conversion
Mr Hugo REGO CAMPELLO
OC28 - Asymmetric Reduction of Enamines towards the Synthesis of (-)-Cytisine and Heterocyclic Building Blocks
Mr Eduardo SANCHEZ
OC16 - Synthesis of Highly Enantioenriched Pyrrolo[1,2-a]Quinolines. Organocatalyzed Domino Cyclopropane Ring Opening/aza-Michael/aldol Reaction Followed by Acid-Promoted Lactamization
Prof. Michael SCHNÜRCH
OC37 - Expansion of the Concept of Nonlinear Effects in Catalytic Reactions Beyond Asymmetric Catalysis
Prof. Henri SCHREKKER
OC30 - Exploring the Antifungal and Antibiofilm Properties of Imidazolium Salts and Fluorescent Benzannulated Benzimidazoles
Mr David Chan Bodin SIEBERT
OC11 - Pyrazoloquinolinones, Revisited GABAA Receptor Tool Compounds
Mr Tim-Daniel J. STUMPF
OC10 - C-Brigded N-Heterocycles as New Ligands
Dr Hiroki TANIMOTO
OC04 - Nitrosoallenes: Reactivity and Applications to Heterocycles Synthesis
Prof. Igor TRUSHKOV
OC24 - Donor-Acceptor Cyclopropanes in Synthesis of Azaheterocycles
Dr Dmitry TSVELIKHOVSKY
OC03 - Rapid Composition of Spiranoid Lactones: Access to Natural and Unexplored Frames
Prof. Jan VAN MAARSEVEEN
OC39 - Methodology Development Towards the Lasso Peptide Series
Dr Esther VICENTE GARCIA
OC26 - Palladium-Catalyzed Isocyanide Insertion in Construction of Diverse Heterocycles
Prof. Guillaume VINCENT
OC34 - Dearomative Arylation of Electrophilic Indoles for the Total Synthesis of Natural Products
Prof. Yanguang WANG
OC23 - 3-Diazoindolin-2-Imines: A Novel Class of Metal Carbene Precursors for the Syntheses of Indole Derivatives
Prof. Daniel B. WERZ
OC18 - Rearrangement and Cycloaddition Reactions of Donor-Acceptor Cyclopropanes