Bioheterocycles 2015

XVI International Conference on Heterocycles in Bioorganic Chemistry

 Metz, France    June 8-11, 2015

Plenary Lectures

PL04 - Non Noble Metal Catalysis for Making Precious Molecules

Prof. Matthias BELLER
Prof. Matthias BELLER
UNIVERSITY OF ROSTOCK, Rostock, Germany
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PL08 - Heterocycles Derived from Natural Products in Management of Multidrug Resistance

Prof. Ahcene BOUMENDJEL
Prof. Ahcene BOUMENDJEL
UNIVERSITÉ JOSEPH FOURIER, Saint-Martin-d'Hčres, France
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PL05 - Metal Catalysis for Heteroarene Synthesis

Prof. Michael GREANEY
Prof. Michael GREANEY
THE UNIVERSITY OF MANCHESTER, Manchester, United Kingdom
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PL06 - The Discovery and Development of the HIV Intergrase Inhibitors Dolutegravir and Cabotegravir

Dr Brian JOHNS
Dr Brian JOHNS
GLAXOSMITHKLINE, NC, United States
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PL07 - Bronsted Acid and Metal-catalyzed Reactions in the Synthesis of Heterocycles

Prof. Esther LETE
Prof. Esther LETE
UNIVERSIDAD DEL PAÍS VASCO, Bilbao, Spain
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PL01 - Photoreactive Heterocycles and Natural Product Derivatives

Prof. Dr Thomas LINDEL
Prof. Dr Thomas LINDEL
TECHNICAL UNIVERSITY OF BRAUNSCHWEIG, Braunschweig, Germany
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PL02 - Targeting DNA Methylation: a Medicinal Chemistry Approach

Prof. Antonello MAI
Prof. Antonello MAI
UNIVERSITY OF ROME "LA SAPIENZA", Rome, Italy
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PL03 - The Importance of Heterocycles in Agrochemistry: Fungicides as a Case Study

Dr Harald WALTER
Dr Harald WALTER
SYNGENTA CROP PROTECTION AG BASEL, Basel, Switzerland
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Invited Lectures

IL07 - Silicon-Containing Tetrahydrocyclopenta[C]Acridine Derivatives as CDKs Inhibitors: Design, Organometallic Synthesis, Metabolic Stability And Optimization

Prof. Philippe BELMONT
Prof. Philippe BELMONT
UNIVERSITY PARIS DESCARTES, Paris, France
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IL01 - Synthetic Explorations in Small-ring Azaheterocyclic Chemistry and Development of Novel Bioactive Heterocycles

Prof. Matthias D'HOOGHE
Prof. Matthias D'HOOGHE
GHENT UNIVERSITY, Ghent, Belgium
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IL09 - Overcoming Resistance with beta-Lactams

Dr Eric DESARBRE
Dr Eric DESARBRE
BASILEA PHARMACEUTICA, Basel, Switzerland
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IL08 - At the Crossroads of Chemistry and Biology: Inhibiting Protein Kinase CK2 by Heterocyclic Small Molecules

Prof. Marc LE BORGNE
Prof. Marc LE BORGNE
UNIVERSITÉ CLAUDE BERNARD LYON 1, Lyon, France
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IL06 - Utilization of Hypervalent Iodonium Reagents for the Construction and Functionalization of Heterocyclic Molecules

Dr Zoltan NOVAK
Dr Zoltan NOVAK
EÖTVÖS UNIVERSITY, Budapest, Hungary
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IL04 - New Methods in Thioamide Chemistry

Dr Mike PORTER
Dr Mike PORTER
UNIVERSITY COLLEGE LONDON, London, United Kingdom
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IL05 - Are Generic Drugs Only a Copy_and_Paste Products?

Prof. Stanislav RADL
Prof. Stanislav RADL
ZENTIVA, Prague, Czech Republic
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IL03 - Synthesis of Novel Alpha7-nAchR Ligands: from an Idea to in Rodent Results for Alzheimer [18F] TEP Imaging

Prof. Sylvain ROUTIER
Prof. Sylvain ROUTIER
UNIVERSITÉ D'ORLÉANS, Orléans, France
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IL02 - Synthesis of Biorelevant Heterocycles with N-heterocyclic Carbenes

Prof. Andreas SCHMIDT
Prof. Andreas SCHMIDT
TECHNICAL UNIVERSITY CLAUSTHAL, Clausthal-Zellerfeld, Germany
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Oral Communications

OC10 - Flavylium-Based Pigments – “Click” Synthesis & Biological Relevance

Dr Stefan CHASSAING
ITAV, Toulouse, France

OC16 - Discovery Of Novel Thieno[3,2-b]Pyrrole 5-Carboxamides as Potent Inhibitors of Chikungunya Virus (CHIKV)

Mr Kuan Chieh CHING
NATIONAL UNIVERSITY OF SINGAPORE, Singapore, Singapore

OC01 - Heterocycle-Peptide Hybrids: Synthesis, Conformational Analysis, and Utilization in Medicinal Chemistry

Mr Luca GENTILUCCI
UNIVERSITA DI BOLOGNA, Bologna, Italy

OC06 - An Original Domino Radical Cyclisation/Smiles Rearrangement Combination: Application to the Synthesis of Indolo[2,3-b]Quinoline-Type Derivatives

Dr. Stéphane GERARD
UNIVERSITÉ DE REIMS - CHAMPAGNE-ARDENNE, REIMS, France

OC05 - Recent Advances in the Total Synthesis of Phormidolides B and C

Mr Alejandro GIL ESCOLANO
IRB BARCELONA, Barcelona, Spain

OC08 - Synthesis of Long Regioregular Dialkyl-Substituted Alpha-Oligofurans

Dr Edward KORSHIN
THE WEIZMANN INSTITUTE OF SCIENCE, Rehovot, Israel

OC15 - Mixed Cu(II) Cu(I) Complexes with Bioheterocycles as the Platform for Construction of Novel Anticancer Agents

Ms Olga KRASNOVSKAYA
MOSCOW STATE UNIVERSITY, Moscow, Russia

OC13 - Synthesis of Imidazo-Pyrrolo-Pyrazines/Diazepines/Diazocines via Domino Ugi/Micheal Reaction and Silver-Catalyzed Heteroannulation

Mr Zhenghua LI
KU LEUVEN, Leuven, Belgium

OC11 - Synthesis of 7-(2-Aminophenyl)- and 7-(4-Aminophenyl)Guanine, DNA Adducts Derived from the Phenylnitrenium Ion

Prof. Igor LINHART
UNIVERSITY OF CHEMISTRY AND TECHNOLOGY, Prague, Czech Republic

OC04 - Novel Cross-Conjugated Dienones Based on 4-Piperidone Moiety: Synthesis and Antitumor Properties

Dr Mikhail MAKAROV
NESMEYANOV INSTITUTE OF ORGANOELEMENT COMPOUNDS OF RAS, Moscow, Russia

OC03 - Diverse Synthesis of Natural Product Inspired Fused and Spiro-Heterocyclic Scaffolds via Ring Distortion And Construction Strategy

Prof. Subhabrata SEN
SHIV NADAR UNIVERSITY, Gautam Budh nagar, India

OC02 - Exploiting the Zincke Reaction to Produce Sophisticated Heptamethine Dyes

Dr Robert SMITH
UNIVERSITY OF CENTRAL LANCASHIRE, Prestoin, United Kingdom

OC07 - Palladium-Catalyzed Cross-Coupling Reactions in the Asymmetric Synthesis of Pyrrolo[1,2-b]Isoquinolines

Prof. Nuria SOTOMAYOR
UNIVERSIDAD DEL PAÍS VASCO / EUSKAL HERRIKO UNIBERTSITATEA, Leioa - Bizkaia, Spain

OC12 - Heterocyclic Coumarine Analogs as Zinc Metalloprotease Inhibitors

Mr Peteris TRAPENCIERIS
LATVIAN INSTITUTE OF ORGANIC SYNTHESIS, RIGA, Latvia