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EFMC 2nd Short Course on Medicinal Chemistry |
| 11/04/2010 |
| 18:00 | Dinner |
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| 19:30 | Introduction to Safety & Attrition Workshop |
Dr Alan STOBIE
(PFIZER, Sandwich, United Kingdom) |
| 21:00 | Close |
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| 12/04/2010 |
| 08:30 | General Overview of Current Safety and Toxicity Testing |
Dr Dominic WILLIAMS
(UNIVERSITY OF LIVERPOOL, Liverpool, United Kingdom) |
| 10:30 | Coffee Break |
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| 11:00 | Small Molecule Based Attrition (1) - Structural 'Alerts' |
Dr Julian BLAGG
(THE INSTITUTE OF CANCER RESEARCH, Surrey, United Kingdom) |
| 12:30 | Lunch |
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| 13:30 | Small Molecule Based Attrition (2) - Molecular Properties |
Dr Julian BLAGG
(THE INSTITUTE OF CANCER RESEARCH, Surrey, United Kingdom) |
| 15:30 | Tea Break |
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| 16:00 | Off-Target Based Attrition (1) - Ion Channel Safety |
Dr Chris POLLARD
(ASTRAZENECA, Macclesfield, United Kingdom) |
| 18:00 | Close |
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| 19:30 | Dinner |
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| 13/04/2010 |
| 08:30 | Off-Target Based Attrition (2) - Role of Transporter Interactions in Toxicology and Attrition |
Dr Gerry KENNA
(ASTRAZENECA, Macclesfield, United Kingdom) |
| 10:00 | Coffee Break |
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| 10:30 | Admet or DMPK Based Attrition |
Dr Don WALKER
(PFIZER, Sandwich, United Kingdom) |
| 12:30 | Lunch |
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| 13:30 | Choosing the Right Target |
Dr Alan STOBIE
(PFIZER, Sandwich, United Kingdom) |
| 13:30 | Attrition (3) - Insilico Prediction Methods |
Dr Alan STOBIE
(PFIZER, Sandwich, United Kingdom) |
| 14:30 | The Safety and Attrition Game |
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| 18:00 | Close |
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| 19:30 | Dinner |
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| 14/04/2010 |
| 08:30 | Newer Methods of Predicting Toxicity (1) - Characterising Mechanisms of Toxicity |
Dr Mark M. GOSINK
(PFIZER, Groton, United States) |
| 10:00 | Coffee Break |
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| 10:30 | Newer Methods of Predicting Toxicity (2) - Use of Whole Cell Invitro Methods |
Dr Jim DYKENS
(PFIZER, Sandwich, United Kingdom) |
| 12:30 | Lunch |
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| 13:30 | Course Ends |
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