XXIIIrd European Colloquium on Heterocyclic Chemistry 09/09/2008
Chairman
Dr Lieven MEERPOEL
19:00 Evening lecture on the life, work and personality of Dr. P. Janssen (founder of Janssen Pharmaceutica).
Dr. Paul J. LEWI
10/09/2008
08:45 Opening Ceremony
Chairman
Prof. Mikael BEGTRUP
09:00 Synthesis of Heterocycles via Alkoxyallenes
Prof. Hans-Ulrich REISSIG
09:50 JNJ-26483327 - A 'Macrocyclic' Multi-Targeted Kinase Inhibitor in Phase I Clinical Trials for the Treatment of Cancer
Dr. Eddy FREYNE
10:20 Ring Transformations and Peculiar Reactions of Functionalized β-Lactams
Prof. Norbert DE KIMPE
11:10 Coffee
11:40 Oral Communications - Session 1
Chairmen
Dr Koen VAN AKEN (ECOSYNTH, Oostende, Belgium) Prof. Christian STEVENS (UGENT, Ghent, Belgium) Prof. Kourosch ABBASPOUR TEHRANI (VUB/UA, Brussels/Antwerp, Belgium)
(R1) (R2) (R3)
Synthesis and Cytotoxicity Evaluation of New Aziridine Containing Benzimidazolequinones
Dr. Fawaz ALDABBAGH
Addition of Organometallics to Cyclic Nitrones: Key Step for the Synthesis of Potent Inhibitors of Alpha-L-Fucosidases
Ms Amélie CASTIGLIA
Application of Microwave-Irradiation as Efficient and Green Reaction Conditions for Various Cycloadditions of 2H -Pyran-2-ones
Dr Kristof KRANJC
Synthesis and Properties of New Fluorophores with a Pyrimidine Central Unit
Prof Georges DUPAS
Synthesis of New Pyrimido[5,4-d ]Pyrimidinones
Dr Ana Helena BACELAR
Transformations of 3,3-Dichloroazetidines to Alkynylimines via 3-Chloro-2-azetines as Strained Intermediates
Dr Sven MANGELINCKX
Novel Routes towards Arylated Oxazoles and Thiazoles through Regioselective Direct C-H Arylation of Oxazole and Thiazole 4-carboxylate Scaffolds
Dr Christophe HOARAU
Preparation, Structural Studies and Reactivity of 1,2-Diazetidines
Mr Mike BROWN
Functionalized 2,5-Diryridinyl-pyrroles by Electrochemical Reduction of 3,6-Dipyridinyl-pyridazine Precursors
Ms Cécile MARIE
12:35 Lunch
13:20 Poster Session 1
Chairman
Prof. Gyorgy HAJÓS
14:20 Novel Organometallic Routes to Polyheterocyclic Ring Systems of Pharmacological Interest
Prof. Hans-Joachim KNÖLKER
14:50 Versatile Synthesis of Novel Ring-Fused 1,5-Benzodiazepines
Dr. Koen VANDYCK
15:20 Competitive Rearrangements of O-N Bond Containing Azoles: the "Power" of a "Weak" Bond
Prof. Andrea PACE
15:50 Coffee
Chairman
Prof. Dirk TOURWE
16:20 Applications of 3-Amino-2-Piperidones to the Synthesis of Peptidomimetics
Prof. Anna DIEZ
16:50 Making and Breaking Heterocyclic Rings via Metal Catalyzed Reactions
Prof. Mark LAUTENS
17:50 Transportation to the City
20:00 Concert in the Cathedral
11/09/2008
Chairman
Prof. Branko STANOVNIK
09:00 Organocatalytic versus Metal-Catalysed Selective Indole Functionalisation: Just a Matter of Choice?
Prof. Alfredo RICCI
09:50 Novel Synthesis of 2,4-Disubstituted Pyrimidines, Key Intermediates in the Synthesis of HIV Compounds
Dr. Fred STAPPERS
10:20 Synthesis and Properties of Novel (Indolo)carbazole Materials
Prof. Wim DEHAEN
11:10 Coffee
11:40 Oral Communications - Session 2
Chairmen
Prof. Kourosch ABBASPOUR TEHRANI (VUB/UA, Brussels/Antwerp, Belgium) Dr Koen VAN AKEN (ECOSYNTH, Oostende, Belgium) Dr Pieter VAN DER VEKEN (UNIVERSITY OF ANTWERP, Antwerpen, Belgium)
(R1) (R2) (R3)
A New Synthesis of Substituted Pyrrole-2-Carboxylates by a Tandem Sonogashira Coupling 5-Endo-DIG-Cyclization from a beta-Iododehydrophenylalanine and Terminal Alkynes
Dr Agathe BEGOUIN
New Meso-Tetraarylporphyrin Derivatives via N-H Insertion Reactions with Diazo Compounds
Ms Ana Teresa PEIXOTO DE CAMPOS GOMES
Functional Analogues of Tröger's Base: New Synthetic Methods and Facile, Predictable Chromatographic Means for the Separation of Enantiomers
Dr Sergey SERGEYEV
A Regio- and Stereospecific Synthesis of t -4-Amino-3-hydroxy- and t ,t -4-Amino-3,5-dihydroxypiperidines
Dr Igor TRUSHKOV
A Novel Multicomponent Reaction towards Imidazolidine-2-thions
Mr Maurice MOOIJMAN
A Novel Practical Synthesis of Licofelone
Dr Stanislav RADL
Sequential Metal-Catalyzed N-Heteroarylation and C–C Cross-Coupling Reactions: An Expedient Route to Tris (hetero)aryl Systems
Mr Jamie SIDDLE
Toward the Total Synthesis of Enantiomerically Pure Antitumor Agent : TMC-69-6H
Ms Sophie VUONG
Polynitrogen Fused Tricyclic Compounds via a Nitrene-Mediated N-N Bond Formation
Ms Coralie NYFFENEGGER
Monocyclic and Dimeric 1,2,4-Triazines Useful Substrates for the Preparation of New Heterocyclic Systems and Natural Products
Dr Andrzej RYKOWSKI
3+2 Cycloadditions of 3-Pyrazolidinone-1-azomethine Imines: an Easy Access to Polysubstituted Pyrazolo[1,2-a ]pyrazolones
Prof Jurij SVETE
An Efficient Microwave-Assisted Synthesis of Disubstituted 2-Amino-1H -imidazoles
Mr Denis ERMOLATEV
12:55 Lunch
13:40 Poster Session 2
Chairman
Prof. Johan VAN DER EYCKEN
14:40 Recent Developments Employing Heterocycles in Asymmetric Catalysis
Prof. Patrick GUIRY
15:10 Pyrrolidinones and Oxindoles as Templates for the Discovery of Innovative Treatments of Epilepsy
Dr. Laurent TURET
15:40 New Catalytic Reactions Designed for the Efficient Synthesis of Natural Products
Prof. Timothy DONOHOE
16:10 Coffee
Chairman
Prof. Guy QUÉGUINER
16:40 Palladium-Catalyzed Multicomponent and Domino Processes for Syntheses of Heterocycles
Prof. Jieping ZHU
17:10 Quinolones, Bisquinolones and Microwaves
Prof. Oliver KAPPE
18:00 Transportation to the City
12/09/2008
Chairman
Prof. Volker JÄGER
09:00 Selective Introduction of a Nitrogen-Containing Functionality into Organic Molecules
Prof. Slovenko POLANC
09:50 Golden Tools for the Synthesis of Heterocycles
Prof. Stephen HASHMI
10:20 Conferences Announcements
Chairman
Prof. Henk VAN DER PLAS
10:30 SNH Reactions in Heterocycles
Prof. Oleg CHUPAKHIN
11:20 Coffee
Chairman
Dr. Laurent PROVINS
11:50 Novel Indole Chemistry in the Synthesis of Heterocycles
Prof. Gordon GRIBBLE
12:20 Efficient Synthesis of Heterocyclic Natural Products and Materials by Domino Reactions
Prof. Lutz F. TIETZE
12:50 Transportation to the City
15:00 Excursion
20:00 Conference Dinner (De Ark)
13/09/2008
Chairman
Dr. Kristof VAN EMELEN
09:00 π-Extended Tetrathiafulvalenes and Fullerenes: Complementary Topological and Electronic Molecules
Prof. Nazario MARTÍN
09:50 Synthesis of Natural Product Inspired Heterocyclic Compound Libraries
Prof. Floris RUTJES
10:20 Syntheses of Carbocyclic β-Amino Acids via Heterocyclic Intermediates
Prof. Ferenc FÜLOP
11:10 Coffee
Chairman
Prof. Erik VAN DER EYCKEN
11:40 Design and Synthesis of Novel Enzyme Inhibitors. Focus on Microwave-Acceleration and Metal-Catalyzed Transformations
Prof. Mats LARHED
12:30 Mn- and Fe-Catalyzed Coupling Reactions: Recent Advances
Prof. Gérard CAHIEZ
13:20 Annoucement of 24ECHC by Johannes Froehlich
13:30 Closing
13:40 Transportation to the City
<Previous page
